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Amphetamine is known to inhibit monoamine oxidase, whereas the flexibility of amphetamine and its metabolites to inhibit numerous P450 isozymes and also other enzymes has not been adequately elucidated. In vitro experiments with human microsomes indicate minimal inhibition of CYP2D6 by amphetamine and insignificant inhibition of CYP1A2, 2D6, and 3A